Anti Diabetic API

• Appearance
• White to off-white powder

• CAS No
• 842133-18-0

• Chemical Name
• Canagliflozin

• Color
• Other, White to off-white

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• Not more than 0.001%

• Loss on Drying
• Not more than 0.5%

• Medicine Name
• Canagliflozin

• Melting Point
• 119-123C

• Molecular Formula
• C24H25FO5S

• Molecular Weight
• 444.52 g/mol

• Particle Size
• 90% <10 micron

• Physical Form
• Solid

• Poisonous
• Other, Non-poisonous when handled as directed

• Purity(%)
• >=99%

• Shelf Life
• 24 months from date of manufacture

• Smell
• Other, Odorless

• Solubility
• Soluble in DMSO and methanol, slightly soluble in water

• Storage
• Other, Store in tightly closed container, at 2-8C, protected from light and moisture

• Structural Formula
• Available upon request

• Type
• Other, Active Pharmaceutical Ingredient (API)

• Usage
• Used for the treatment of type 2 diabetes mellitus

• Appearance
• White to off-white powder

• Boiling point
• Not applicable (decomposes before boiling)

• CAS No
• 960404-48-2

• Chemical Name
• Dapagliflozin propanediol monohydrate

• Color
• White

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• 0.001%

• Loss on Drying
• 1.0%

• Medicine Name
• Dapagliflozin

• Melting Point
• 126-128C

• Molecular Formula
• C21H25ClO6

• Molecular Weight
• 408.87 g/mol

• Particle Size
• D90 < 150 microns

• Ph Level
• 5.0 - 7.0 (1% solution)

• Physical Form
• Solid

• Poisonous
• Other, Non-poisonous if used as intended

• Purity(%)
• >= 99.0%

• Shelf Life
• 36 months

• Smell
• Other, Odorless

• Solubility
• Slightly soluble in water, soluble in methanol and ethanol

• Storage
• Other, Store in a cool, dry place, protect from light

• Structural Formula
• Available on request

• Taste
• Bitter

• Type
• Other, Active Pharmaceutical Ingredient (API)

• Usage
• Used for the treatment of Type 2 Diabetes Mellitus

• Appearance
• White to off-white powder

• Boiling point
• Not applicable (decomposes)

• CAS No
• 668270-12-0

• Chemical Name
• 8-[(3R)-3-Amino-1-piperidinyl]-7-(but-2-yn-1-yl)-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]-3,7-dihydro-1H-purine-2,6-dione

• Color
• Other, White to off-white

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• Not more than 0.001%

• Loss on Drying
• Not more than 0.5%

• Medicine Name
• Linagliptin

• Melting Point
• > 200C

• Molecular Formula
• C25H28N8O2

• Molecular Weight
• 472.54 g/mol

• Particle Size
• D90 < 10 microns

• Ph Level
• 6.0 - 7.5 (1% w/v solution)

• Physical Form
• Solid

• Poisonous
• NO

• Purity(%)
• >= 99.0

• Shelf Life
• 3 years

• Smell
• Other, Odorless

• Solubility
• Sparingly soluble in water; freely soluble in dimethyl sulfoxide (DMSO) and methanol

• Storage
• Other, Store in a cool, dry place, tightly closed container

• Structural Formula
• Available on request

• Type
• Other, Active Pharmaceutical Ingredient (API)

• Usage
• Used in the treatment of type 2 diabetes mellitus

• Appearance
• White to off-white powder

• CAS No
• 361442-04-8

• Chemical Name
• (1S,3S,5S)-2-[(2S)-2-Amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile

• Color
• Other, White to off-white

• EINECS No
• 681-803-0

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• NMT 0.001%

• Loss on Drying
• NMT 0.5%

• Medicine Name
• Saxagliptin

• Melting Point
• >200C

• Molecular Formula
• C18H25N3O2

• Molecular Weight
• 315.41 g/mol

• Particle Size
• D90 <10 microns

• Physical Form
• Solid

• Poisonous
• NO

• Purity(%)
• >=99%

• Shelf Life
• 24 months

• Smell
• Other, Odorless

• Solubility
• Soluble in DMSO, slightly soluble in water

• Storage
• Other, Store in a cool, dry place, protected from light

• Structural Formula
• Refer to image

• Taste
• Bitter

• Type
• Other, Active Pharmaceutical Ingredient

• Usage
• Used in the treatment of type 2 diabetes mellitus

• Appearance
• White or off-white powder

• Boiling point
• Not applicable (decomposes)

• CAS No
• 654671-77-9

• Chemical Name
• Sitagliptin Phosphate Monohydrate

• Color
• Other, White to off-white

• EINECS No
• 698-872-8

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• NMT 0.001%

• Loss on Drying
• NMT 0.5%

• Medicine Name
• Sitagliptin

• Melting Point
• 206-210C

• Molecular Formula
• C16H15F6N5OH3PO4H2O

• Molecular Weight
• 523.32 g/mol

• Particle Size
• D90 NMT 150 microns

• Ph Level
• 4.0 - 6.0 (1% w/v aqueous solution)

• Physical Form
• Powder

• Poisonous
• NO

• Purity(%)
• >= 99%

• Shelf Life
• 36 months

• Smell
• Other, Odorless

• Solubility
• Soluble in water, slightly soluble in methanol

• Storage
• Other, Store in a cool, dry place, tightly closed, away from heat and light

• Structural Formula
• Available on request

• Taste
• Bitter

• Type
• Other, Active Pharmaceutical Ingredient

• Usage
• Anti-diabetic medication, used for the treatment of type 2 diabetes mellitus

• Appearance
• White to off-white crystalline powder

• CAS No
• 274901-16-5

• Chemical Name
• (S)-1-[(3-Hydroxy-1-adamantyl)amino]acetyl-2-cyanopyrrolidine

• Color
• Other, White to off-white

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• Not more than 0.001%

• Loss on Drying
• Not more than 0.5%

• Medicine Name
• Vildagliptin Active Pharmaceutical Ingredients

• Melting Point
• 146-150C

• Molecular Formula
• C17H25N3O2

• Molecular Weight
• 303.40 g/mol

• Particle Size
• Typically D90 <10 microns

• Ph Level
• Neutral

• Physical Form
• Solid

• Poisonous
• Other, No (used under medical supervision)

• Purity(%)
• 99.0%

• Shelf Life
• 36 months from date of manufacture

• Smell
• Other, Odorless

• Solubility
• Soluble in methanol, slightly soluble in water

• Storage
• Other, Store in a cool, dry, and well-ventilated place, protected from light

• Structural Formula
• C17H25N3O2 (Skeletal structure available upon request)

• Taste
• Bitter

• Type
• Other, API (Active Pharmaceutical Ingredient)

• Usage
• Used as an antidiabetic agent in the treatment of type 2 diabetes mellitus

• Appearance
• White or almost white crystalline powder

• Boiling point
• Not applicable (decomposes)

• CAS No
• 21187-98-4

• Chemical Name
• 1-(hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-3-methylsulfonylurea

• Color
• White

• EINECS No
• 244-482-5

• Grade
• Other, Pharmaceutical Grade

• HS Code
• 29420090

• Heavy Metal (%)
• 0.001%

• Loss on Drying
• Not more than 0.5%

• Medicine Name
• Gliclazide

• Melting Point
• 165-170C

• Molecular Formula
• C15H21N3O3S

• Molecular Weight
• 323.41 g/mol

• Particle Size
• Not more than 10 micron

• Physical Form
• Solid

• Poisonous
• NO

• Purity(%)
• 99%

• Shelf Life
• 3 years

• Smell
• Other, Odorless

• Solubility
• Practically insoluble in water; freely soluble in acetone; sparingly soluble in ethanol

• Storage
• Other, Store in a cool, dry place, protected from light

• Structural Formula
• C15H21N3O3S

• Taste
• Bitter

• Type
• Other, Active Pharmaceutical Ingredient

• Usage
• Used for the treatment of type 2 diabetes mellitus